KR-31831 improves survival and protects hematopoietic cells and radiosensitive tissues against radiation-induced injuries in mice. Biomedicine & Pharmacotherapy. Vol.146, 112350. (2022.02.01)
PredMS: a random Forest model for predicting metabolic stability of drug candidates in human liver microsomes. Bioinformatics. Vol. 38, 364-368. (2022.01.15.)
Identification of new target proteins of a Urotensin-II receptor antagonist using transcriptome-based drug repositioning approach. Scientific Reports. Vol.11, 17138. (2021.08.24.)
KR-39038, a novel GRK5 inhibitor, attenuates cardiac hypertrophy and improves cardiac function in heart failure. Biomolecules & Therapeutics. Vol. 28, 482-489 (2020.08.29.)
DeepHIT: a deep learning framework for prediction of hERG-induced cardiotoxicity. Bioinformatics. Vol. 36, 3049-3055. (2020.05.15.)
Optimization of cyclic sulfamide derivatives as 11beta-hydroxysteroid dehydrogenase 1 inhibitors for the potential treatment of ischemic brain injury. Bioorganic & Medicinal Chemistry Letters. Vol. 30, 126787. (2020.01.15.)
Icariin protects against radiation-induced mortality and damage in vitro and in vivo.
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DITMD-induced mitotic defects and apoptosis in tumor cells by blocking the polo-box domain-dependent functions of polo-like kinase 1. European Journal of Pharmacology. Vol. 847. 113-122. (2019.03.15)